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As a GLP-1 receptor agonist, it works by mimicking the natural incretin hormone GLP-1 to increase insulin secretion in a glucose-dependent manner, suppress glucagon release, slow gastric emptying by approximately 35%, and reduce appetite through central nervous system signaling

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Harris, Triple-Hormone Combination Retatrutide Induces 24% Body Weight Loss, JAMA, vol

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When taken at the recommended dosage, GLP-1s can cause unwanted side effects, like nausea, GI issues, and dizziness

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Front Endocrinol (Lausanne) 2022;13:1043789

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Available from: Hall KD, Kahan S

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These fibers reach the colon where they are fermented by gut bacteria into butyrate

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