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Importantly, methylated esters of TCA intermediates, such as DMF, are cell permeable and can modify the activity of this pathway by increasing the level of metabolic intermediates' proximate to fumarate

Pancreatitis was reported as a rare serious adverse event in clinical trials

The most direct human safety study involved only 2 healthy participants, which is far too small to rule out uncommon side effects, long-term risks, injection-related complications, or product-quality concerns
Bowers et al
